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GT 949
CAS No. 460330-27-2
GT 949 ( —— )
产品货号. M26706 CAS No. 460330-27-2
GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥518 | 有现货 |
|
| 10MG | ￥915 | 有现货 |
|
| 25MG | ￥1847 | 有现货 |
|
| 50MG | ￥3345 | 有现货 |
|
| 100MG | ￥5006 | 有现货 |
|
| 500MG | ￥10773 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称GT 949
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).
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产品描述GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).(In Vitro):GT 949 displays selectivity to EAAT2 and has no effect on glutamate activity mediated by EAAT1 or EAAT3. GT 949 improves glutamate transport (EC50 = 0.26 nM) and increases glutamate transport in a non-competitive manner with an increase in Vmax of about 47% in EAAT2-transfected cells.
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同义词——
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通路Others
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靶点Other Targets
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受体5-HT; Dopamine
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研究领域——
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适应症——
化学信息
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CAS Number460330-27-2
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分子量527.7
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分子式C30H37N7O2
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纯度>98% (HPLC)
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溶解度——
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SMILESCOc1ccc2[nH]c(=O)c(cc2c1)C(N1CCN(CC1)C1CCCCC1)c1nnnn1CCc1ccccc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Shan-Meng Lin, et al. Structure-Based Stabilization of Non-native Protein-Protein Interactions of Coronavirus Nucleocapsid Proteins in Antiviral Drug Design. J Med Chem. 2020 Mar 26;63(6):3131-3141.
产品手册
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